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质量水平
检测方案
≥95.0%
形式
solid
mp
289-293 °C
SMILES字符串
CS(=O)(=O)c1ccc(cc1)B(O)O
InChI
1S/C7H9BO4S/c1-13(11,12)7-4-2-6(3-5-7)8(9)10/h2-5,9-10H,1H3
InChI key
VDUKDQTYMWUSAC-UHFFFAOYSA-N
一般描述
含不定量的酸酐
应用
4-(甲磺酰基)苯硼酸可作为试剂用于以下反应：
试剂用于制备
- Suzuki交叉偶联反应
- 铜催化芳基硼酸的氧化三氟甲基硫醇化反应
- 3-溴呋喃及相关杂环的定向金属化和区域选择性官能化反应
- Barton-Zard吡咯环缩合和Baeyer-Villiger氧化反应
- 二聚体环加成和钯催化的交叉偶联过程
- 用于奥当卡替中间体合成的连续流Suzuki反应
试剂用于制备
- 二芳基氨基吡啶类化合物，可作为潜在抗疟药
- 氢吡喃并吡嗪，通过氯吡嗪甲醛和烯化反应
- 联芳基砜衍生物，作为组胺H3受体的拮抗剂
- 具有潜在抗肿瘤作用的新型激酶抑制剂支架
- N-羟基异喹啉的丙型肝炎病毒抑制活性
用于 4-氧代丁烯酰胺的铑催化不对称 1,4-加成的高效硼酸。
WGK
WGK 3
闪点(°F)
Not applicable
闪点(°C)
Not applicable
Copper-catalyzed oxidative trifluoromethylthiolation of aryl boronic acids with TMSCF3 and elemental sulfur.
Chao Chen et al.
Angewandte Chemie (International ed. in English), 51(10), 2492-2495 (2012-01-31)
Pamela Kassis et al.
European journal of medicinal chemistry, 46(11), 5416-5434 (2011-09-29)
We here report the synthesis and biological evaluation of new 3-[(2-indolyl)]-5-phenyl-3,5-pyridine, 3-[(2-indolyl)]-5-phenyl-2,4-pyridine and 3-[(2-indolyl)]-5-phenyl-2,6-pyrazine derivatives designed as potential CDK inhibitors. Indoles and phenyls were used to generate several substitutions of the pyridine and pyrazine rings. The synthesis included Stille or
Synthesis of 2,6-disubstituted-7,8-dihydro-6H-pyrano[2,3-b]pyrazines
Li, J-C.; et al.
Tetrahedron Letters, 53, 852-853 (2012)
Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-(2-(4'-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine (APD916)
Semple, G.; et al.
Bioorganic & Medicinal Chemistry, 21, 71-75 (2012)
Yue-Lei Chen et al.
Bioorganic & medicinal chemistry, 20(1), 467-479 (2011-11-22)
C7-Substituted 2-hydroxyisoquinoline-1,3-diones inhibit the strand transfer of HIV integrase (IN) and the reverse-transcriptase-associated ribonuclease H (RNH). Hepatitis C virus (HCV) NS5B polymerase shares a similar active site fold to RNH and IN, suggesting that N-hydroxyimides could be useful inhibitor scaffolds
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