生物来源
synthetic (organic)
质量水平
检测方案
≥98% (TLC)
形式
powder
效能
636 nM Ki
溶解性
DMSO: soluble (Dilute in aqueous medium immediately prior to use and store on ice for no more than 12 hours.)
degassed ethanol: soluble (Dilute in aqueous medium immediately prior to use and store on ice for no more than 12 hours.)
λmax
224 nm
储存温度
−20°C
SMILES字符串
[H]\C(Br)=C1\CCC(C(=O)O1)c2cccc3ccccc23
InChI
1S/C16H13BrO2/c17-10-12-8-9-15(16(18)19-12)14-7-3-5-11-4-1-2-6-13(11)14/h1-7,10,15H,8-9H2/b12-10+
InChI key
BYUCSFWXCMTYOI-ZRDIBKRKSA-N
生化/生理作用
来自P388D巨噬细胞(IC 50 = 8μM)的钙取代磷脂酶A2和镁取代磷脂酸磷酸磷酸酶的强效,不可逆抑制剂;酶激活的不可逆糜蛋白酶抑制剂(K i = 636 nM)。
WGK
WGK 3
个人防护装备
dust mask type N95 (US), Eyeshields, Gloves
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商品
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