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  • Acyl sulfonamide anti-proliferatives. Part 2: activity of heterocyclic sulfonamide derivatives.

Acyl sulfonamide anti-proliferatives. Part 2: activity of heterocyclic sulfonamide derivatives.

Bioorganic & medicinal chemistry letters (2005-01-25)
Mary M Mader, Chuan Shih, Eileen Considine, Alfonso De Dios, Cora Sue Grossman, Philip A Hipskind, Ho-Shen Lin, Karen L Lobb, Beatriz Lopez, José E Lopez, Luisa M Martin Cabrejas, Michael E Richett, Wesley T White, Yiu-Yin Cheung, Zhongping Huang, John E Reilly, Sean R Dinn
摘要

The anti-proliferative activity of acylated heterocyclic sulfonamides is described in Vascular Endothelial Growth Factor-dependent Human Umbilical Vascular Endothelial Cells (VEGF-HUVEC) and in HCT116 tumor cells in a soft agar diffusion assay.