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444244

MMP-2 Inhibitor I

Name: MMP-2 Inhibitor I
Brand: MM

The MMP-2 Inhibitor I, also referenced under CAS 10335-69-0, controls the biological activity of MMP-2. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.

Synonym(s):

MMP-2 Inhibitor I, cis-9-Octadecenoyl-N-hydroxylamide, Oleoyl-N-hydroxylamide, OA-Hy

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About This Item

Empirical Formula (Hill Notation):

C₁₈H₃₅NO₂

CAS Number:

10335-69-0

Molecular Weight:

297.48

UNSPSC Code:

12352200

NACRES:

NA.77

Quality Level

100

Assay

≥98% (HPLC)

form

solid

potency

1.7 mM K_i

manufacturer/tradename

Calbiochem^®

storage condition

OK to freeze
protect from light

color

white

solubility

DMSO: 2 mg/mL
ethanol: 3 mg/mL

shipped in

wet ice

storage temp.

−20°C

InChI

1S/C18H35NO2/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-16-17-18(20)19-21/h9-10,21H,2-8,11-17H2,1H3,(H,19,20)/b10-9-

InChI key

LTXHELLMCCEDJG-KTKRTIGZSA-N

General description

A cell-permeable, potent inhibitor of MMP-2 that acts in a dose-dependent manner (K_i = 1.7 µM).

Potent inhibitor of MMP-2 (gelatinase A). Inhibits MMP-2 in a dose dependent manner (K_i = 1.7 µM)

Biochem/physiol Actions

Cell permeable: yes

Primary Target
MMP-2

Product does not compete with ATP.

Reversible: no

Packaging

Packaged under inert gas

Warning

Toxicity: Standard Handling (A)

Reconstitution

Unstable in solution; reconstitute just prior to use.

Other Notes

Berton, A., et. al. 2001. J. Biol. Chem.276, 20458.
Emonard, H., et al. 1999. Ann. N.Y. Acad. Sci.878, 647.

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

WGK

WGK 1

Flash Point(F)

Not applicable

Flash Point(C)

Not applicable

Certificates of Analysis (COA)

Search for Certificates of Analysis (COA) by entering the products Lot/Batch Number. Lot and Batch Numbers can be found on a product’s label following the words ‘Lot’ or ‘Batch’.

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