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质量水平
检测方案
>98% (HPLC)
形式
solid
颜色
white
溶解性
DMSO: >10 mg/mL
H2O: insoluble
创始人
Sanofi Aventis
SMILES字符串
Cc1c(nn(-c2ccc(Cl)cc2Cl)c1-c3ccc(I)cc3)C(=O)NN4CCCCC4
InChI
1S/C22H21Cl2IN4O/c1-14-20(22(30)27-28-11-3-2-4-12-28)26-29(19-10-7-16(23)13-18(19)24)21(14)15-5-8-17(25)9-6-15/h5-10,13H,2-4,11-12H2,1H3,(H,27,30)
InChI key
BUZAJRPLUGXRAB-UHFFFAOYSA-N
基因信息
mouse ... Cnr1(12801) , Cnr2(12802)
rat ... Cnr1(25248)
应用
AM251，一种CB1 大麻素受体拮抗剂，已被用于一项研究，以确定其与海马神经元的相互作用，以增强小鼠的空间记忆。
生化/生理作用
AM251是一种CB1 大麻素受体拮抗剂。
特点和优势
该化合物由Sanofi Aventis开发。要浏览其他药物开发化合物和批准的药物/候选药物列表，单击此处。
其他说明
盐含量可能会有所不同。
危险声明
预防措施声明
危险分类
Aquatic Chronic 4
WGK
WGK 3
闪点(°F)
Not applicable
闪点(°C)
Not applicable
个人防护装备
dust mask type N95 (US), Eyeshields, Gloves
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